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Ein fluoreszenzmarkiertes Physalaemin-Analoges mit hoher biologischer Aktivität

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Summary

The synthesis of fluorescent labelled derivative of the N-terminal physalaemin hexapeptide [6–11], which contains a 1-dimethylaminoaphtalene-5-sulfonyl residue at the α-amino group of the N-terminal Lysine, is described. Pharmacological data of the fluorescent labelled compound as compared with the unsubstituted peptide are reported.

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Authors and Affiliations

  1. Institut für Pharmakologie, Deutsche Akademie der Wissenschaften zu Berlin, 1115, Berlin-Buch, DDR

    B. Mehlis, H. Apelt, J. Bergmann, H. Niedrich & P. Oehme

Authors
  1. B. Mehlis
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  2. H. Apelt
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  3. J. Bergmann
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  4. H. Niedrich
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  5. P. Oehme
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Mehlis, B., Apelt, H., Bergmann, J. et al. Ein fluoreszenzmarkiertes Physalaemin-Analoges mit hoher biologischer Aktivität. Experientia 27, 930–931 (1971). https://doi.org/10.1007/BF02135751

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  • DOI: https://doi.org/10.1007/BF02135751

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