Abstract
Selective methods for deriving 1′-aryl-, 1′-indolyl-, 1′-pyrrolyl- and 1′-methyl-substituted 3-vinylindoles2 are described. In all cases the precursors were 3-acylindoles. The new compounds are synthetically useful synthons for annelation of the indole skeleton.
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Pindur, U., Pfeuffer, L. Selektive Synthesen zu 1′-aryl-, 1′-hetaryl-und 1′-alkylsubstituierten 3-Vinylindolen. Monatsh Chem 118, 1031–1038 (1987). https://doi.org/10.1007/BF00815329
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DOI: https://doi.org/10.1007/BF00815329