Derivatives of β-casomorphins with high analgesic potency
References (39)
- et al.
A superactive antinociceptive pentapeptide, (D-Met2, Pro5)-enkephalinamide
FEBS Lett
(1977) - et al.
Opioid activities of β-casomorphins
Life Sci
(1981) - et al.
Antinociceptive potencies of β-casomorphin analogs as compared to their affinity towards μ and δ-opiate receptor sites in brain and periphery
Peptides
(1982) - et al.
Participation of both ‘enkephalinase’ and aminopeptidase activities in the metabolism of endogenous enkephalins
Neuroscience
(1983) - et al.
Evidence for analgesic activity of β-casomorphin in rats
Neurosci Lett
(1981) - et al.
Naloxazone irreversibly inhibits the high affinity binding of (125J) D-Ala-D-Leu5-enkephalin
Life Sci
(1981) - et al.
β-Casomorphins—novel opioid peptides derived from bovine caseine—isolation and structure
- et al.
Structure-activity relationship of orally active enkephalins analogues as analgesics
Life Sci
(1979) - et al.
Development of opiate tolerance/dependence in the guinea-pig myenteric plexus and the mouse vas deferens
- et al.
Are there subtypes (isoreceptors) of multiple opiate receptors in the mouse vas deferens?
Eur J Pharmacol
(1981)
Biological inactivation of enkephalins and the role of enkephalin-carboxypeptidase (‘enkephalinase’) as neuropeptidase
Life Sci
(1981)
A differential interaction of putative μ-selective agonists with opiate binding sites in rat brain
Neurochem Intern
(1982)
Minimum structure opioids—Dipeptide and tripeptide analogs of the enkephalins
Peptides
(1981)
Post-proline cleaving enzyme. Synthesis of a new fluorogenic substrate and distribution of the endopeptidasein rat tissues and body fluids of man
Biochim Biophys Acta
(1979)
Mu and delta receptors: Correlation with high and low affinity opiate binding sites
Eur J Pharmacol
(1980)
The actions of naloxazone on the binding and analgesic properties of morphiceptin (NH2-Tyr-Pro-Phe-Pro-CONH2), a selective mu receptor ligand
Life Sci
(1981)
Drug-receptor interaction: Interaction of one or more drugs with one receptor system
Morphiceptin (NH2-Tyr-Pro-Phe-Pro-CONH2): A potent and specific agonist for morphine (μ) receptors
Science
(1981)
Analgesic activity of intracerebroventricular administration of morphiceptin and β-casomorphins: Correlation with the morphin (μ) receptor binding affinity
Life Sci
(1982)
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